An efficient synthesis of N-protected β-aminoethanesulfonyl chlorides: versatile building blocks for the synthesis of oligopeptidosulfonamides

AJ Brouwer, MCF Monnee, RMJ Liskamp

Index: Synthesis, , # 11 p. 1579 - 1584

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Citation Number: 38

Abstract

... Originally, peptidosulfon- amides were synthesized by the reaction of a b-amino ... Using these Fmoc-protected aminoethanesulfonyl chlorides, we were able to synthesize oligopeptidosulfonamides on the ... for solid phase synthesis, because the efficiency of the synthesis ...