A three-step synthesis of 4-(4-iodo-1H-pyrazol-1-yl) piperidine, a key intermediate in the synthesis of Crizotinib
SJ Fussell, A Luan, P Peach, G Scotney
Index: Tetrahedron Letters, , vol. 53, # 8 p. 948 - 951
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Citation Number: 5
Abstract
... Tetrahedron Letters. Volume 53, Issue 8, 22 February 2012, Pages 948–951. ... Koning, Andrew Derrick, Alan Happe, and Asayuki Kamatani for useful discussions and support throughout the project; Stuart Green, Hayley Jackman, and Stewart Hayes for the support of this Letter. ...
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