Tetrahedron Letters

One-pot N-alkylation/Heck approach to substituted indoles

ML Weinrich, HP Beck

Index: Weinrich, Melissa L.; Beck, Hilary P. Tetrahedron Letters, 2009 , vol. 50, # 50 p. 6968 - 6972

Full Text: HTML

Citation Number: 19

Abstract

Due to the prevalence of indole functionality in several biologically active molecules, many research efforts are focused on developing novel general, mild, and efficient methods for the regioselective preparation of substituted indoles from readily available starting materials. 1 The intramolecular Heck reaction has been widely used for the synthesis of substituted indoles. 2 In addition, indoles have been prepared utilizing one-pot cascade reactions. 3 For example, the palladium- ...

Related Articles:

Enamine Rearrangement of Pyridinium Salts to Indole Ring: A Combined Experimental and Molecular Modeling Study

[Hosaan, Aisha; Fadda, Ahmed A. Journal of Heterocyclic Chemistry, 2013 , vol. 50, # 3 p. 638 - 644]

Regioselective Hydroarylation Reactions of C3 Electrophilic N??Acetylindoles Activated by FeCl3: An Entry to 3??(Hetero) arylindolines

[Beaud, Rodolphe; Guillot, Regis; Kouklovsky, Cyrille; Vincent, Guillaume Chemistry - A European Journal, 2014 , vol. 20, # 24 p. 7492 - 7500]

Regioselective Hydroarylation Reactions of C3 Electrophilic N??Acetylindoles Activated by FeCl3: An Entry to 3??(Hetero) arylindolines

[Beaud, Rodolphe; Guillot, Regis; Kouklovsky, Cyrille; Vincent, Guillaume Chemistry - A European Journal, 2014 , vol. 20, # 24 p. 7492 - 7500]

Regioselective Hydroarylation Reactions of C3 Electrophilic N??Acetylindoles Activated by FeCl3: An Entry to 3??(Hetero) arylindolines

[Beaud, Rodolphe; Guillot, Regis; Kouklovsky, Cyrille; Vincent, Guillaume Chemistry - A European Journal, 2014 , vol. 20, # 24 p. 7492 - 7500]

Regioselective Hydroarylation Reactions of C3 Electrophilic N??Acetylindoles Activated by FeCl3: An Entry to 3??(Hetero) arylindolines

[Beaud, Rodolphe; Guillot, Regis; Kouklovsky, Cyrille; Vincent, Guillaume Chemistry - A European Journal, 2014 , vol. 20, # 24 p. 7492 - 7500]

More Articles...