Pyrazolo [1, 5-a] pyrimidines, triazolo [1, 5-a] pyrimidines and their tricyclic derivatives as corticotropin-releasing factor 1 (CRF 1) receptor antagonists
T Saito, T Obitsu, C Minamoto, T Sugiura…
Index: Bioorganic and Medicinal Chemistry, , vol. 19, # 20 p. 5955 - 5966
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Citation Number: 21
Abstract
... Bioorganic & Medicinal Chemistry. ... Significant contributions have been made in the past two decades by several pharmaceutical research groups to discover non-peptide CRF 1 receptor antagonists as a potential treatment for stress-related illnesses (including depression). ...
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[Saito, Tetsuji; Obitsu, Tetsuo; Minamoto, Chiaki; Sugiura, Tsuneyuki; Matsumura, Naoya; Ueno, Sonoko; Kishi, Akihiro; Katsumata, Seishi; Nakai, Hisao; Toda, Masaaki Bioorganic and Medicinal Chemistry, 2011 , vol. 19, # 20 p. 5955 - 5966]