A general synthesis of dioxolenone prodrug moieties

CQ Sun, PTW Cheng, J Stevenson, T Dejneka…

Index: Tetrahedron Letters, , vol. 43, # 7 p. 1161 - 1164

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Citation Number: 22

Abstract

... Tetrahedron Letters. Volume 43, Issue 7, 11 February 2002, Pages 1161–1164. ... presumably occurs via the initial O-acylation intermediate 5, then undergoes enolization and subsequent cyclization to afford 6. Hydrogenolysis of benzyl ester 6 provided the acid 7, which was ...

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