Modulators of the human CCR5 receptor. Part 2: SAR of substituted 1-(3, 3-diphenylpropyl)-piperidinyl phenylacetamides

…, S McLaughlin, J Oldfield, JS Shaw, H Tucker…

Index: Cumming, John G.; Cooper, Anne E.; Grime, Ken; Logan, Chris J.; McLaughlin, Sharon; Oldfield, John; Shaw, John S.; Tucker, Howard; Winter, Jon; Whittaker, David Bioorganic and Medicinal Chemistry Letters, 2005 , vol. 15, # 22 p. 5012 - 5015

Full Text: HTML

Citation Number: 29

Abstract

Download PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... SAR and DMPK studies led to the identification of substituted N-alkyl-N-[1-(3,3-diphenylpropyl)piperidin -4-yl]-2-phenylacetamides as potent and orally bioavailable ligands for the human CCR5 chemokine receptor. ... SAR and DMPK studies led to the identification of substituted N-alkyl-N-[1-(3, ...

Related Articles:

Efficient and Mild Iron-Catalyzed Direct Allylation of Benzyl Alcohols and Benzyl Halides with Allyltrimethylsilane

[Han, Jie; Cui, Zili; Wang, Jianguo; Liu, Zhongquan Synthetic Communications, 2010 , vol. 40, # 14 p. 2042 - 2046]

Iterative molecular assembly based on the cation-pool method. Convergent synthesis of dendritic molecules

[Okajima, Masayuki; Soga, Kazuya; Nokami, Toshiki; Suga, Seiji; Yoshida, Jun-Ichi Organic Letters, 2006 , vol. 8, # 22 p. 5005 - 5007]

Iterative molecular assembly based on the cation-pool method. Convergent synthesis of dendritic molecules

[Okajima, Masayuki; Soga, Kazuya; Nokami, Toshiki; Suga, Seiji; Yoshida, Jun-Ichi Organic Letters, 2006 , vol. 8, # 22 p. 5005 - 5007]

Iterative molecular assembly based on the cation-pool method. Convergent synthesis of dendritic molecules

[Okajima, Masayuki; Soga, Kazuya; Nokami, Toshiki; Suga, Seiji; Yoshida, Jun-Ichi Organic Letters, 2006 , vol. 8, # 22 p. 5005 - 5007]

Generation of Diarylcarbenium Ion Pools via Electrochemical CH Bond Dissociation

[Okajima, Masayuki; Soga, Kazuya; Watanabe, Takashi; Terao, Kimitada; Nokami, Toshiki; Suga, Seiji; Yoshida, Jun-Ichi Bulletin of the Chemical Society of Japan, 2009 , vol. 82, # 5 p. 594 - 599]

More Articles...