Chemoselective cyclocondensation of α-acylacetamidines with 2-methylsulfanyl-4, 6-dichloropyrimidine-5-carbaldehyde

SG Ryazanov, SI Selivanov, DV Dar'in…

Index: Ryazanov; Selivanov; Dar'in; Lobanov; Potekhin Russian Journal of Organic Chemistry, 2008 , vol. 44, # 2 p. 288 - 291

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Citation Number: 5

Abstract

Abstract Cyclocondensation of α-acylacetamidine with 2-methylsulfanyl-4, 6- dichloropyrimidine-5-carbaldehyde proceeds chemo-and regioselectively involving replacement by the α-carbon of the amidine of the chlorine in the aromatic ring and a reaction of the amino group with the formyl group.