Discovery, Modeling, and Human Pharmacokinetics of N-(2-Acetyl-4, 6-dimethylphenyl)-3-(3, 4-dimethylisoxazol-5-ylsulfamoyl) thiophene-2-carboxamide (TBC3711), …
C Wu, ER Decker, N Blok, H Bui, TJ You…
Index: Journal of Medicinal Chemistry, , vol. 47, # 8 p. 1969 - 1986
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Citation Number: 105
Abstract
... Journal of Medicinal Chemistry. ... 12-14. The potentially wide application of endothelin antagonists has spurred intensive medicinal research and a number of chemical entities are being evaluated in the clinic. ... Synthetic Chemistry. ...
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