Multisubstrate inhibition of 4-hydroxybenzoate 3-monooxygenase

FG Salituro, DA Demeter, HJR Weintraub…

Index: Salituro; Demeter; Weintraub; Lippert; Resvick; McDonald Journal of Medicinal Chemistry, 1994 , vol. 37, # 24 p. 4076 - 4078

Full Text: HTML

Citation Number: 4

Abstract

4-Hydroxybenzoate 3-monooxygenase (p-hydroxybenzoate hydroxylase, PHBH; EC 1.14. 13.21, isolated from Pseudomonas fluorescens, is a very well-characterized NADPH- dependent flavin-mono~ xygenasel-~ which catalyzes the conversion of p-hydroxybenzoate to 3, 4-dihydroxybenzoate (Scheme 1). Extensive enzyme kinetics, 6 inhibition studie~,~-~ and X-ray crystallographic studieslnJ1 have been published. The enzyme mechanism has ...

Related Articles:

Flavonoid metabolism: the synthesis of phenolic glucuronides and sulfates as candidate metabolites for bioactivity studies of dietary flavonoids

[Zhang, Qingzhi; Raheem, K. Saki; Botting, Nigel P.; Slawin, Alexandra M.Z.; Kay, Colin D.; O'Hagan, David Tetrahedron, 2012 , vol. 68, # 22 p. 4194 - 4201]

New aromatic inhibitors of EPSP synthase incorporating hydroxymalonates as novel 3-phosphate replacements

[Shah, Ajit; Font, Jose L.; Miller, Michael J.; Ream, Joel E.; Walker, Mark C.; Sikorski, James A. Bioorganic and Medicinal Chemistry, 1997 , vol. 5, # 2 p. 323 - 334]

Flavonoid metabolism: the synthesis of phenolic glucuronides and sulfates as candidate metabolites for bioactivity studies of dietary flavonoids

[Zhang, Qingzhi; Raheem, K. Saki; Botting, Nigel P.; Slawin, Alexandra M.Z.; Kay, Colin D.; O'Hagan, David Tetrahedron, 2012 , vol. 68, # 22 p. 4194 - 4201]

Flavonoid metabolism: the synthesis of phenolic glucuronides and sulfates as candidate metabolites for bioactivity studies of dietary flavonoids

[Zhang, Qingzhi; Raheem, K. Saki; Botting, Nigel P.; Slawin, Alexandra M.Z.; Kay, Colin D.; O'Hagan, David Tetrahedron, 2012 , vol. 68, # 22 p. 4194 - 4201]

More Articles...