The optimization of aminooxadiazoles as orally active inhibitors of Cdc7
PE Harrington, MP Bourbeau, C Fotsch, M Frohn…
Index: Bioorganic and Medicinal Chemistry Letters, , vol. 23, # 23 p. 6396 - 6400
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Citation Number: 5
Abstract
... Bioorganic & Medicinal Chemistry Letters. ... a Medicinal Chemistry, Amgen Inc., One Amgen Center Drive, Thousand Oaks, CA 91320, USA; ... The chemical matter leading to 1 was identified through high throughput screening of analogs from our protein kinase B (PKB) program. ...
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