A new class of potent non-imidazole H 3 antagonists: 2-aminoethylbenzofurans
M Cowart, JK Pratt, AO Stewart, YL Bennani…
Index: Bioorganic and Medicinal Chemistry Letters, , vol. 14, # 3 p. 689 - 693
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Citation Number: 83
Abstract
... Bioorganic & Medicinal Chemistry Letters. Volume 14, Issue 3, 9 February 2004, Pages 689–693. ... However, in spite of the likely medical utility of H 3 antagonists, no agent in the class has yet received clinical approval, perhaps due to inadequate drug-like properties. ...
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A new class of potent non-imidazole H 3 antagonists: 2-aminoethylbenzofurans
[Cowart, Marlon; Pratt, John K.; Stewart, Andrew O.; Bennani, Youssef L.; Esbenshade, Timothy A.; Hancock, Arthur A. Bioorganic and Medicinal Chemistry Letters, 2004 , vol. 14, # 3 p. 689 - 693]
[Angewandte Chemie - International Edition, , vol. 51, # 6 p. 1405 - 1407]