Structure–activity relationships of diamine inhibitors of cytochrome P450 (CYP) 3A as novel pharmacoenhancers, part I: Core region

H Liu, L Xu, H Hui, R Vivian, C Callebaut…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 24, # 3 p. 989 - 994

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Abstract

... Bioorganic & Medicinal Chemistry Letters. ... a Department of Medicinal Chemistry, Gilead Sciences, Foster City, CA, USA; b Department of Drug Metabolism, Gilead Sciences ... of Biology, Gilead Sciences, Foster City, CA, USA; d Department of Structural Chemistry, Gilead Sciences ...

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