[125I] Iodoproxyfan and related compounds: a reversible radioligand and novel classes of antagonists with high affinity and selectivity for the histamine H3 receptor

H Stark, K Purand, A Hüls, X Ligneau…

Index: Journal of medicinal chemistry, , vol. 39, # 6 p. 1220 - 1226

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Citation Number: 77

Abstract

... Journal of Medicinal Chemistry. ... Chemistry. The key synthetic intermediate of all H 3 receptor antagonists of the new series is 3-(1H-imidazol-4-yl)propanol (3). This compound could be prepared starting from urocanic ...

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