Synthesis of 2-amino-4-pyrimidinones from resin-bound guanidines prepared using bis (allyloxycarbonyl)-protected triflylguanidine
CW Zapf, M Goodman
Index: Alberola, Angel; Antolin, Luis F.; Gonzalez, Ana M.; Laguna, Miguel A.; Pulido, Francisco J. Heterocycles, 1987 , vol. 25, p. 393 - 397
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Citation Number: 18
Abstract
... J. Org. ... 7,8 With these findings, attempts were undertaken to synthesize heterocycles from resin-bound guanidines 31 and 32 using β-keto esters ... was the best solvent (Table 1) for the clean conversion of the resin-bound guanidine 31 into the corresponding heterocycle utilizing β ...
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