Palladium??Catalyzed DYKAT of Butadiene Monoepoxide: Enantioselective Total Synthesis of (+)??DMDP,(−)??Bulgecinine, and (+)??Broussonetine G

…, DB Horne, MJ Woltering

Index: Trost, Barry M.; Horne, Daniel B.; Woltering, Michael J. Chemistry - A European Journal, 2006 , vol. 12, # 25 p. 6607 - 6620

Full Text: HTML

Citation Number: 100

Abstract

Abstract Palladium catalyzed asymmetric allylic alkylation reaction of an amine with two equivalents of butadiene monoxide allows for the expedient synthesis of trans-and cis-2, 5- dihydropyrroles. The versatility of these chiral synthons towards the synthesis of a wide variety of iminosugar natural products was demonstrated with the short and high yielding asymmetric syntheses of (+)-DMDP, and (−)-bulgecinine. In addition, the first total ...

Related Articles:

Synthesis of 2 (R), 5 (R)-bis (hydroxymethyl)-3 (R), 4 (R)-dihydroxypyrrolidine. A novel glycosidase inhibitor

[Card, Peter J.; Hitz, William D. Journal of Organic Chemistry, 1985 , vol. 50, # 6 p. 891 - 893]

… -α-D-mamnofuranoside as a divergent intermediate for the synthesis of polyhydroxylated piperidines and pyrrolidines: synthesis of 2, 5-dideoxy-2, 5-imino-D-mannitol …

[Fleet, George W. J.; Smith, Paul W. Tetrahedron, 1987 , vol. 43, # 5 p. 971 - 978]

Diastereoselective concise syntheses of the polyhydroxylated alkaloids DMDP and DAB

[Bouillon, Marc E.; Pyne, Stephen G. Tetrahedron Letters, 2014 , vol. 55, # 2 p. 475 - 478]

Synthesis of azasugars as potent inhibitors of glycosidases

[Le Merrer, Yves; Poitout, Lydie; Depezay, Jean-Claude; Dosbaa, Isabelle; Geoffroy, Sabine; Foglietti, Marie-Jose Bioorganic and Medicinal Chemistry, 1997 , vol. 5, # 3 p. 519 - 533]

Intramolecular benzyl protection delivery: A practical synthesis of DMDP and DGDP from D-fructose

[Organic Letters, , vol. 8, # 2 p. 297 - 299]

More Articles...