Oxaziridine??Mediated Oxyamination of Indoles: An Approach to 3??Aminoindoles and Enantiomerically Enriched 3??Aminopyrroloindolines

T Benkovics, IA Guzei, TP Yoon

Index: Benkovics, Tamas; Guzei, Ilia A.; Yoon, Tehshik P. Angewandte Chemie - International Edition, 2010 , vol. 49, # 48 p. 9153 - 9157

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Citation Number: 62

Abstract

Pyrroloindoline natural products have attracted considerable interest because of both their biological activity and their unique structures.[1] Nature presumably produces these architecturally fascinating compounds through electrophilic cyclization cascades involving appropriately functionalized tryptamine and tryptophan precursors. In the laboratory, the use of chemical oxidants (eg, m-chloroperbenzoic acid, dioxirane, N-bromosuccinimide) to ...

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