Journal of heterocyclic chemistry

Synthesis of the 1, 2, 3, 4??tetrahydrobenzofuro [2, 3??c] pyridine ring system

JC Jaen, LD Wise

Index: Jaen, Juan C.; Wise, Lawrence D. Journal of Heterocyclic Chemistry, 1987 , vol. 24, p. 1317 - 1319

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Citation Number: 6

Abstract

Abstract As part of an on-going research project, we required an efficient method for the preparation of compounds containing the 1, 2, 3, 4-tetrahydrobenzofuro [2, 3-c] pyridine ring nucleus. The parent compound 1 has not been described in the literature, and there is only one reference to the N-methyl analog 2 [1]. A series of structurally related compounds, the 2- substituted-4-hydroxy-1, 2, 3, 4-tetrahydrobenzofuro [2, 3-c] pyridines, has been described ...

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