Topical carbonic anhydrase inhibitors

RD Schoenwald, MG Eller, JA Dixson…

Index: Schoenwald; Eller; Dixson; Barfknecht Journal of Medicinal Chemistry, 1984 , vol. 27, # 6 p. 810 - 812

Full Text: HTML

Citation Number: 36

Abstract

Discussion Our approach to the development of a topically effective carbonic anhydrase inhibitor involves selecting a suitable prototype molecule, making single molecular modifications of that structure, determining various physical and biological properties of each analogue, and finally utilizing the data to design a molecule with the best combination of properties. When 1 is applied topically to the eye it is inactive. In ow initial studies, we ...

Related Articles:

Improved Synthesis of 2??(3H) Benzothiazolethiones under Microwave Irradiation

[Huang, Wei; Tan, Ying; Ding, Ming-Wu; Yang, Guang-Fu Synthetic Communications, 2007 , vol. 37, # 3 p. 369 - 376]

Synthesis and Biological Evaluation of 2??Mercapto??1, 3??benzothiazole Derivatives with Potential Antimicrobial Activity

[Franchini, Carlo; Muraglia, Marilena; Corbo, Filomena; Florio, Marco Antonio; Di Mola, Antonia; Rosato, Antonio; Matucci, Rosanna; Nesi, Marta; Van Bambeke, Francoise; Vitali, Cesare Archiv der Pharmazie, 2009 , vol. 342, # 10 p. 605 - 613]

More Articles...