The preparation and SAR of 4-(anilino), 4-(phenoxy), and 4-(thiophenoxy)-quinazolines: inhibitors of p56 lck and EGF-R tyrosine kinase activity

MR Myers, NN Setzer, AP Spada, AL Zulli…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 7, # 4 p. 417 - 420

Full Text: HTML

Citation Number: 68

Abstract

... Please enable JavaScript to use all the features on this page. Bioorganic & Medicinal Chemistry Letters. Volume 7, Issue 4, 18 February 1997, Pages 417–420. Cover image Cover image. ... of Medicinal Chemistry Rhône-Poulenc Rorer Pharmaceuticals, 500 Arcola Rd. ...

Related Articles:

(E)-3-(4-oxo-4H-quinazolin-3-yl)-2-propenoic acids, a new series of antiallergy agents

[LeMahieu; Carson; Nason; Parrish; Welton; Baruth; Yaremko Journal of Medicinal Chemistry, 1983 , vol. 26, # 3 p. 420 - 425]

Inhibition studies on Mycobacterium tuberculosis N-acetylglucosamine-1-phosphate uridyltransferase (GlmU)

[Tran, Anh Thu; Wen, Daying; West, Nicholas P.; Baker, Edward N.; Britton, Warwick J.; Payne, Richard J. Organic and Biomolecular Chemistry, 2013 , vol. 11, # 46 p. 8113 - 8126]

Identification of potent and selective inhibitors of PDGF receptor autophosphorylation

[Furuta, Takayuki; Sakai, Teruyuki; Senga, Terufumi; Osawa, Tatsushi; Kubo, Kazuo; Shimizu, Toshiyuki; Suzuki, Rika; Yoshino, Tetsuya; Endo, Megumi; Miwa, Atsushi Journal of Medicinal Chemistry, 2006 , vol. 49, # 7 p. 2186 - 2192]

A novel approach to quinazolin-4 (3H)-one via quinazoline oxidation: an improved synthesis of 4-anilinoquinazolines

[Marzaro, Giovanni; Guiotto, Adriano; Pastorini, Giovanni; Chilin, Adriana Tetrahedron, 2010 , vol. 66, # 4 p. 962 - 968]

Phenylarsonic acid compounds with broad-spectrum and potent cytotoxic activity against human cancer cells

[Arzneimittel-Forschung/Drug Research, , vol. 53, # 6 p. 428 - 439]

More Articles...