Optimisation of two-photon induced cleavage of molecular linker systems for drug delivery

T Buckup, A Southan, HC Kim, N Hampp…

Index: Buckup; Southan; Kim; Hampp; Motzkus Journal of Photochemistry and Photobiology A: Chemistry, 2010 , vol. 210, # 2-3 p. 188 - 192

Full Text: HTML

Citation Number: 6

Abstract

Photoreactive linker systems for drug delivery in modern ophthalmology are crucial for the efficiency of such applications. We compare 5 different linker molecule candidates (truxillic acid and 4 dimers of coumarin derivates) in solution regarding their chemical stability and two-photon induced cleavage efficiency, and shed light into the role of molecular structure in the cleavage reaction. Dimers of the coumarin family showed much higher two-photon ...

Related Articles:

Pivalase catalytic antibodies: towards abzymatic activation of prodrugs

[Bensel, Nicolas; Reymond, Martine T.; Reymond, Jean-Louis Chemistry - A European Journal, 2001 , vol. 7, # 21 p. 4604 - 4612]

7, 8-Disubstituted-but not 6, 7-disubstituted coumarins selectively inhibit the transmembrane, tumor-associated carbonic anhydrase isoforms IX and XII over the …

[Maresca, Alfonso; Scozzafava, Andrea; Supuran, Claudiu T. Bioorganic and Medicinal Chemistry Letters, 2010 , vol. 20, # 24 p. 7255 - 7258]

The behavior of certain coumarins and furocoumarins toward sulfur reagents

[Ibrahim, Nabila Phosphorus, Sulfur and Silicon and the Related Elements, 2006 , vol. 181, # 8 p. 1773 - 1784]

More Articles...