Copper??Catalyzed Synthesis of 4??Aryl??1H??1, 2, 3??triazoles from 1, 1??Dibromoalkenes and Sodium Azide

X Wang, C Kuang, Q Yang

Index: Wang, Xiaokun; Kuang, Chunxiang; Yang, Qing European Journal of Organic Chemistry, 2012 , # 2 p. 424 - 428

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Citation Number: 10

Abstract

Abstract A new methodology for the Cu-catalyzed synthesis of 1H-1, 2, 3-triazoles from 1, 1- dibromoalkenes and sodium azide is presented. Aryl dibromoolefins were efficiently converted into the corresponding 1, 2, 3-triazoles. A comprehensive number of functional groups were compatible with this reaction. 1, 2, 3-Triazoles were obtained in moderate to excellent yields.

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