Modulation on C??and N??Terminal Moieties of a Series of Potent and Selective Linear Tachykinin NK2 Receptor Antagonists

M Gensini, M Altamura, T Dimoulas, V Fedi…

Index: ChemMedChem, , vol. 5, # 1 p. 65 - 78

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Citation Number: 5

Abstract

... ChemMedChem, 5: 65–78. ... Volume: Issue: Page: ... Bromination of naphthalene-2-carboxylic acid 9 with bromine in hot glacial acetic acid gave a mixture of monobromo derivatives from which the 5-bromo-naphthalene-2-carboxylic acid 10 was isolated by crystallization.11. ...