Benefits of a Dual Chemical and Physical Activation: Direct aza-Michael Addition of Anilines Promoted by Solvent Effect under High Pressure

…, J Maddaluno, AY Rulev, J Legros

Index: Lebleu, Thomas; Ma, Xiaolu; Maddaluno, Jacques; Legros, Julien Chemical Communications, 2014 , vol. 50, # 15 p. 1836 - 1838

Full Text: HTML

Citation Number: 4

Abstract

The unique combination of hexafluoroisopropanol (HFIP) employed as solvent and hyperbaric conditions (10–15 kbar) allows unprecedented 1, 4-addition of poor nucleophiles, such as aromatic amines, onto sluggish (cumbersome) Michael acceptors

Related Articles:

A convenient 1, 3-dipolar cycloaddition–reduction synthetic sequence from 2-allyloxy-5-nitro-salicylaldehyde to aminobenzopyran-annulated heterocycles

[Parmar, Narsidas J.; Pansuriya, Bhavesh R.; Labana, Balvantsingh M.; Kant, Rajni; Gupta, Vivek K. RSC Advances, 2013 , vol. 3, # 38 p. 17527 - 17539]

Microwave-Assisted Synthesis of Substituted Hexahydro-pyrrolo [3, 2-c] quinolines

[Neuschl, Michal; Bogdal, Darek; Potacek, Milan Molecules, 2007 , vol. 12, # 1 p. 49 - 59]

More Articles...