S-[2-(. omega.-Aminoalkylamino) ethyl] dihydrogen phosphorothioates and related compounds as potential antiradiation agents
JR Piper, CR Stringfellow Jr, RD Elliott…
Index: Piper,J.R. et al. Journal of Medicinal Chemistry, 1969 , vol. 12, # 2 p. 236 - 243
Full Text: HTML
Citation Number: 82
Abstract
011 known aziridine intermediates. 6 These beginnings, marked by a high level of activity, were then expanded into a series of homologs and analogs. The two routes that led to the S- 2-(w-aminoalkylamino) ethyl dihydrogen phosphorothioates 3 are outlined in Scheme I; one involved the Cortese conversion'of hydroxyethylated cqw-alkanediamines, and the other involved the Gabriel synthesis from intermediates made available by the recently developed
Related Articles:
[Kong, Yu; Tan, Rong; Zhao, Lili; Yin, Donghong Green Chemistry, 2013 , vol. 15, # 9 p. 2422 - 2433]
[Henig, Joerg; Mamedov, Ilgar; Fouskova, Petra; Toth, Eva; Logothetis, Nikos K.; Angelovski, Goran; Mayer, Hermann A. Inorganic Chemistry, 2011 , vol. 50, # 14 p. 6472 - 6481]
[Hamer; Rathbone Journal of the Chemical Society, 1943 , p. 243,247]