Tricyclic indole-2-carboxylic acids: highly in vivo active and selective antagonists for the glycine binding site of the NMDA receptor

S Katayama, N Ae, T Kodo, S Masumoto…

Index: Journal of Medicinal Chemistry, , vol. 46, # 5 p. 691 - 701

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Citation Number: 30

Abstract

... Journal of Medicinal Chemistry. ... Chemistry. Tricyclic indole-2-carboxylic acid derivatives (3) bearing various anilide groups can be prepared by condensation of tricyclic indole monocarboxylic acid 3S-(−)-4 with the ...

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