Synthesis of a glycosylated ortho-carboranyl amino acid
C Thimon, L Panza, C Morin
Index: Thimon, Christian; Panza, Luigi; Morin, Christophe Synlett, 2003 , # 10 p. 1399 - 1402
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Citation Number: 9
Abstract
Abstract The preparation of an ortho-carborane derivative bearing both carbohydrate and amino acid substituents is presented; opening of a glucofuranuro-γ-lactone derivative with propargylamines, cycloaddition of decaborane to an acetylenic bond and amidation with a N- Fmoc-glutamate derivative are the key-steps in this synthesis.
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