A CONVENIENT SYNTHESIS OF NEW HALOTHIENYL β-AMINOACIDS AS VERSATILE BUILDING BLOCKS

O Renault, P Dallemagne, S Rault

Index: Renault, Olivier; Dallemagne, Patrick; Rault, Sylvain Organic Preparations and Procedures International, 1997 , vol. 29, # 4 p. 488 - 494

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Citation Number: 3

Abstract

During the course of our work on the synthesis of new thiophene derivatives with therapeutic interest,',* we needed reasonable quantities of new P-aminoacids which are versatile building-blocks in heterocyclic chemistry and in the synthesis of peptid0mimetics.'-'We previously reported the preparation and the chemical reactivity of several P-amino-P- arylpropionic acid derivatives (Scheme I)."'" The present work describes the multigram ...