Molecules
Synthesis and Biological Evaluation of Thieno [3, 2-d]-pyrimidinones, Thieno [3, 2-d] pyrimidines and Quinazolinones: Conformationally Restricted 17b- …
E Perspicace, S Marchais-Oberwinkler, RW Hartmann
Index: Molecules, , vol. 18, # 4 p. 4487 - 4509
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Citation Number: 3
Abstract
... Rigidification is an often applied method to increase the potency of active molecules. ... The condensation of molecule 6 with N,N-dimethylformamide dimethyl acetal (DMF-DMA) gave methyl 3-dimethyl ... The injection volume was 15 µL and flow rate was set to 800 µL/min. ...
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