Efflux inhibitor-1 structure
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Common Name | Efflux inhibitor-1 | ||
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CAS Number | 1776055-29-8 | Molecular Weight | 479.53 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C28H25N5O3 | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of Efflux inhibitor-1Efflux inhibitor-1 (compound 2) is a pyrazolo[1,5-a]pyrimidine efflux inhibitor. Efflux inhibitor-1 selectively targets toward ABCG2/BCRP over ABCB1 with IC50s of 0.45 μM and 2.17 μM, respectively[1]. |
Name | Efflux inhibitor-1 |
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Description | Efflux inhibitor-1 (compound 2) is a pyrazolo[1,5-a]pyrimidine efflux inhibitor. Efflux inhibitor-1 selectively targets toward ABCG2/BCRP over ABCB1 with IC50s of 0.45 μM and 2.17 μM, respectively[1]. |
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Related Catalog | |
Target |
IC50: 0.45 μM (ABCG2/BCRP), 2.17 μM (ABCB1)[1] |
References |
Molecular Formula | C28H25N5O3 |
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Molecular Weight | 479.53 |