PROTAC ERRα ligand 2
Modify Date: 2025-09-11 17:17:00
PROTAC ERRα ligand 2 structure
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Common Name | PROTAC ERRα ligand 2 | ||
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| CAS Number | 2306388-57-6 | Molecular Weight | 445.31 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C20H13F6NO4 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of PROTAC ERRα ligand 2PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist with an IC50 of 5.67 nM. PROTAC ERRα ligand 2 (IC50=5.67 nM) displays a ~11-fold improved potency than XCT790 (IC50=61.3 nM)[1]. |
| Name | PROTAC ERRα ligand 2 |
|---|
| Description | PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist with an IC50 of 5.67 nM. PROTAC ERRα ligand 2 (IC50=5.67 nM) displays a ~11-fold improved potency than XCT790 (IC50=61.3 nM)[1]. |
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| Related Catalog | |
| References |
| Molecular Formula | C20H13F6NO4 |
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| Molecular Weight | 445.31 |
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Name: Ratio of IC50 for XCT790 to IC50 for test compound for binding affinity to GST-tagged...
Source: ChEMBL
Target: Steroid hormone receptor ERR1
External Id: CHEMBL4305575
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Name: Binding affinity to GST-tagged ERRalpha-LBD (unknown origin) using fluorescein-conjug...
Source: ChEMBL
Target: Steroid hormone receptor ERR1
External Id: CHEMBL4305574
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