Synthesis and evaluation of aniline headgroups for alkynyl thienopyrimidine dual EGFR/ErbB-2 kinase inhibitors

AG Waterson, KG Petrov, KR Hornberger…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 19, # 5 p. 1332 - 1336

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Citation Number: 30

Abstract

... JavaScript is disabled on your browser. Please enable JavaScript to use all the features on this page. Bioorganic & Medicinal Chemistry Letters. Volume 19, Issue 5, 1 March 2009, Pages 1332–1336. ... Keywords. Kinase inhibitor; EGFR; ErbB-2; Medicinal chemistry. ...