… /palladium-catalyzed Suzuki–Miyaura coupling of heteroaryl halides with 3-pyridine-and 3-thiopheneboronic acid: an efficient catalyst for the formation of biheteroaryls

K Wang, Q Fu, R Zhou, X Zheng, H Fu…

Index: Wang, Kun; Fu, Qi; Zhou, Rong; Zheng, Xueli; Fu, Haiyan; Chen, Hua; Li, Ruixiang Applied Organometallic Chemistry, 2013 , vol. 27, # 4 p. 232 - 238

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Citation Number: 9

Abstract

Heteroaryls are ubiquitous in biologically active compounds.[1–4] However, for electronic or poisoning reasons, they are not good reactants.[5–7] Palladium-catalyzed Suzuki–Miyaura coupling is a powerful and synthetically valuable process for the preparation of heteroaryl derivatives.[8–11] In recent years, much work has been directed toward the coupling of arylboronic acids with heteroaryl halides,[12–16] but the reactions involving ...