Tetrahedron letters

A facile protocol for the convenient preparation of amino-substituted α-bromo-and α, α-dibromo arylmethylketones

Z Diwu, C Beachdel, DH Klaubert

Index: Diwu, Zhenjun; Beachdel, Christopher; Klaubert, Dieter H. Tetrahedron Letters, 1998 , vol. 39, # 28 p. 4987 - 4990

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Citation Number: 67

Abstract

Download full text in PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... Amino-substituted arylmethylketones are selectively brorninated in sulfuric acid to afford the corresponding dibromomethylarylketones that are then debrominated with diethylphosphite to give the desired bromomethylarylketones in excellent yield. ... The 1 HNMR (CDCl 3 ) ...