Aryl tetrahydropyridine inhibitors of farnesyltransferase: glycine, phenylalanine and histidine derivatives

SL Gwaltney, SJ O'Connor, LTJ Nelson…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 13, # 7 p. 1359 - 1362

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Citation Number: 23

Abstract

... Bioorganic & Medicinal Chemistry Letters. Volume 13, Issue 7, 7 April 2003, Pages 1359–1362. Cover image Cover image. ... We then examined analogues derived from histidine (Scheme 7). Again, much the same chemistry was used for this work. ...

Biarylaniline phenethanolamines as potent and selective β3 a...

[Uehling, David E.; Shearer, Barry G.; Donaldson, Kelly H.; Chao, Esther Y.; Deaton, David N.; Adkison, Kim K.; Brown, Kathleen K.; Cariello, Neal F.; Faison, Walter L.; Lancaster, Mary E.; Lin, Jasmine; Hart, Robert; Milliken, Tula O.; Paulik, Mark A.; Sherman, Bryan W.; Sugg, Elizabeth E.; Cowan, Conrad Journal of Medicinal Chemistry, 2006 , vol. 49, # 9 p. 2758 - 2771]

Application of Organolithium Compounds in Organic Synthesis....

[Synthetic Communications, , vol. 27, # 6 p. 1075 - 1086]