e.g. Filippa Pettersson or Cancer Res. 75(6) , 1102-12, (2015) or 10.1002/anie.201600521
Two-step phosphorus-mediated substitution of hydroxy groups in selected primary alcohols for fluorinated alkyl or aryl substituents: the molecular structure of 1, 1-bis ( …
In an Arbuzov type reaction, amido phosphites (Et2N) 2-PORand a broad range of halofluoro organic halides (X= Cl, Br) formed the corresponding alkylated derivatives R1–R2 [R1= Bn, R2= C (SO2F) 3, CCl2F, CCl2CF3, CBr2F, C (CF3) 3, C6F5; R1= Et, CH2CF3, Me, R2= CCl2CF3], whereas with FC (SO2F) 3 and loss of SO2, BnCF (SO2F) 2 was obtained, as shown by X-ray crystallography.