Discovery of pyrazolthiazoles as novel and potent inhibitors of bacterial gyrase

SM Ronkin, M Badia, S Bellon, AL Grillot…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 20, # 9 p. 2828 - 2831

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Citation Number: 48

Abstract

... Bioorganic & Medicinal Chemistry Letters. ... However, the N-linked piperidine compounds (3b and other substituted N-linked piperidines not shown) were also found to possess chemical stability issues limiting their usefulness. ...