Discovery of novel 2-(aminoheteroaryl)-thiazole-5-carboxamides as potent and orally active Src-family kinase p56 Lck inhibitors

P Chen, D Norris, J Das, SH Spergel, J Wityak…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 14, # 24 p. 6061 - 6066

Full Text: HTML

Citation Number: 34

Abstract

... JavaScript is disabled on your browser. Please enable JavaScript to use all the features on this page. Bioorganic & Medicinal Chemistry Letters. ... Chemistry, Bristol-Myers Squibb Pharmaceutical Research Institute, PO Box 4000, Princeton, NJ 08543-4000, USA; ...

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