Structure-based design of potent and selective 3-phosphoinositide-dependent kinase-1 (PDK1) inhibitors

JR Medina, CJ Becker, CW Blackledge…

Index: Journal of Medicinal Chemistry, , vol. 54, # 6 p. 1871 - 1895

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Citation Number: 28

Abstract

... Journal of Medicinal Chemistry. ... Chem. , 2011, 54 (6), pp 1871–1895. DOI: 10.1021/jm101527u. Publication Date (Web): February 22, 2011. Copyright © 2011 American Chemical Society. *Phone: 610-917-5889. Fax: 610-917-4206. E-mail: jesus.r.medina@gsk.com. †. ...