Tetrahedron letters

Aziridination of alkenes by 3-amino-2-ethylquinazolin-3H-4-one and lead tetra-acetate-trifluoroacetic acid

RS Atkinson, CM Darrah, BJ Kelly

Index: Atkinson, Robert S.; Darrah, Christine M.; Kelly, Brian J. Tetrahedron Letters, 1987 , vol. 28, # 15 p. 1711 - 1712

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Citation Number: 9

Abstract

... AEIRIDINATION OF ALKENES BY 3-AMINO-2-ETHYLQUIN.AEOLIN-3~-4-ONE AND Robert S. (Department of LEAD TBTRA-ACETATE-TRIFLUOROACETIC ACID Atkinson*, Christine M. Darrah, and Brian J. Kelly Chemistry, Leicester University, LeiCeSter LB1 7RH, UK) SUMMARY : A number of alkenes undergo aziridination in good yield by oxidative addition of the title N-aminoquinazolone (1) only in the presence of TFA. ...