Synthesis and fungicidal activity of novel 1, 3??disubstituted 1H??diazirine derivatives

…, LV Shahbazyan, SV Harutyunyan…

Index: Eliazyan, Karine A.; Avetisyan, Frunze V.; Jivanshiryan, Tamara L.; Pivazyan, Vergush A.; Ghazaryan, Emma A.; Shahbazyan, Lusya V.; Harutyunyan, Siranush V.; Yengoyan, Aleksandr P. Journal of Heterocyclic Chemistry, 2011 , vol. 48, # 1 p. 118 - 123

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Citation Number: 2

Abstract

Abstract A convenient method for synthesis of novel 1-[pyrimidinyl], 1-[1, 3, 5-triazin-2- carbonyl], and 1-[thiazol-5-carbonyl] derivatives of 3-thioxo-diaziridine 1, 3, 5, and 7 from corresponding hydrazides, CS2, and KOH is elaborated. The highest reaction yield was observed when these initial reagents were taken in molar ratio of 1: 1.7: 2.0, respectively. By alkylation of compounds 1, 3, 5, and 7 that proceeds exclusively at sulfur atom, the 3- ...