Synthesis

Solvent-free Heck-Jeffery reactions under ball-milling conditions applied to the synthesis of unnatural amino acids precursors and indoles

E Tullberg, F Schacher, D Peters, T Frejd

Index: Synthesis, , # 7 p. 1183 - 1189

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Citation Number: 31

Abstract

... This methodology provides a useful and direct synthesis of some of these derivatives. ... [12] Some of the tested amino- or hydroxyl-substituted aryl iodides were commercially available: 3, 5, 6, 9, 10, 20 and 29; others: 1, 2, 4, 7, 22 and 30 were synthesized according to ...