Affinity and activity profiling of unichiral 8-substituted 1, 4-benzodioxane analogues of WB4101 reveals a potent and selective α 1B-adrenoceptor antagonist

L Fumagalli, M Pallavicini, R Budriesi, M Gobbi…

Index: European Journal of Medicinal Chemistry, , vol. 58, p. 184 - 191

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Citation Number: 8

Abstract

... European Journal of Medicinal Chemistry. Volume 58, December 2012, Pages 184–191. Cover image Cover image. Original article. ... (i) H 2 –Pd/C, MeOH. (j) K 2 CO 3 , acetone. (k) 2-(2,6-Dimethoxyphenoxy)ethylamine, isobutanol; HCl/EtOH. ...