Total synthesis of (8R)-3-(2-deoxy-. beta.-D-erythro-pentofuranosyl)-3, 6, 7, 8-tetrahydroimidazo [4, 5-d][1, 3] diazepin-8-ol (pentostatin), the potent inhibitor of …

E Chan, SR Putt, HDH Showalter…

Index: Journal of Organic Chemistry, , vol. 47, # 18 p. 3457 - 3464

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Citation Number: 58

Abstract

... US. Patent 3030376) by the procedure described by: Allsebrook, WE; Gulland, J. M.; Story, LF J. Chem. SOC. 1942,232. ... Therefore, the following chemistry was carried out (using conditions as for the analogous reactions in the Experimental Section). ...