3-(Indol-2-yl) indazoles as Chek1 kinase inhibitors: Optimization of potency and selectivity via substitution at C6

ME Fraley, JT Steen, EJ Brnardic, KL Arrington…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 16, # 23 p. 6049 - 6053

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Citation Number: 42

Abstract

... Please enable JavaScript to use all the features on this page. Bioorganic & Medicinal Chemistry Letters. ... Department of Medicinal Chemistry, Merck Research Laboratories, West Point, PA 19486, USA; ... American Chemical Society, San Diego, CA, March 2005; Abstract MEDI-121. ...