Palladium??Catalyzed Amination of Aryl Mesylates

…, Z Zhou, CP Lau, FY Kwong

Index: So, Chau Ming; Zhou, Zhongyuan; Lau, Chak Po; Kwong, Fuk Yee Angewandte Chemie - International Edition, 2008 , vol. 47, # 34 p. 6402 - 6406

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Citation Number: 136

Abstract

Palladium-catalyzed C (sp2) ÀN bond-forming reactions have evolved into a highly versatile and synthetically attractive transformation in targeting pharmaceutically useful intermediates.[1] Since the discovery of the first catalytic amination method,[2] efforts have been made toward increasing the reaction efficacy.[3] Notable ligands, such as tBu3P,[4] Beller and co-workers PAP,[5] Buchwald and co-workers biaryl phosphines,[6] Hartwig ...