Novel orally active, dibenzazepinone-based γ-secretase inhibitors

JU Peters, G Galley, H Jacobsen, C Czech…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 17, # 21 p. 5918 - 5923

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Citation Number: 28

Abstract

... JavaScript is disabled on your browser. Please enable JavaScript to use all the features on this page. Bioorganic & Medicinal Chemistry Letters. ... We prepared ∼50 compounds by parallel chemistry, most of which were inactive and often had low microsomal stabilities. ...