Preparation and bioevaluation of 99mTc nitrido radiopharmaceuticals with pyrazolo [1, 5-a] pyrimidine as tumor imaging agents

…, H Liu, X Wang, M Feng, C Qi, J Zhang, C Peng

Index: Ding, Rui; He, Yong; Xu, Jingli; Liu, Hang; Wang, Xiao; Feng, Man; Qi, Chuanmin; Zhang, Junbo; Peng, Cheng Medicinal Chemistry Research, 2012 , vol. 21, # 4 p. 523 - 530

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Citation Number: 12

Abstract

Abstract The 7-(2-aminoethylamino)-5-methyl-3-cyanopyrazolo [1, 5-a] pyrimidine (AMCPP) was synthesized and conjugated with N-mercaptoacetylglycine (MAG), N- mercaptoacetylphenylalanine (MAF), and N-mercaptoacetylvaline (MAA), respectively. ...