Tetrahedron letters

N-Alkylation of 1H-indoles and 9H-carbazoles with alcohols

A Bombrun, G Casi

Index: Bombrun, Agnes; Casi, Giulio Tetrahedron Letters, 2002 , vol. 43, # 12 p. 2187 - 2190

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Citation Number: 32

Abstract

A comparative study of N-alkylation of 1H-indole and 9H-carbazole derivatives with alcohol derivatives was performed using classic Mitsunobu reaction conditions, ie DEAD/PPh3, azodicarboxamide derivatives such as TMAD in the presence of PBu3, or using phosphorane derivatives such as CMMP.