Discovery of a potent, selective and orally active canine COX-2 inhibitor, 2-(3-difluoromethyl-5-phenyl-pyrazol-1-yl)-5-methanesulfonyl-pyridine

J Li, KML DeMello, H Cheng, SM Sakya…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 14, # 1 p. 95 - 98

Full Text: HTML

Citation Number: 38

Abstract

... Bioorganic & Medicinal Chemistry Letters. ... Veterinary Medicine Research and Development, Pfizer Inc., Groton, CT 06340, USA. Received 7 July 2003, Revised 30 September 2003, Accepted 5 October 2003, Available online 13 November 2003. Abstract. ...