Discovery of N-{1-[3-(3-oxo-2, 3-dihydrobenzo [1, 4] oxazin-4-yl) propyl] piperidin-4-yl}-2-phenylacetamide (Lu AE51090): an allosteric muscarinic M1 receptor agonist …

AG Sams, M Hentzer, GK Mikkelsen…

Index: Journal of Medicinal Chemistry, , vol. 53, # 17 p. 6386 - 6397

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Citation Number: 24

Abstract

... Journal of Medicinal ... Medicinal Chemistry Research. ‡ Molecular Pharmacology. § Discovery ADME. ∥ In Vivo Neuropharmacology. Lundbeck Research Denmark, H ... During the 1990s, several pharmaceutical companies pursued selective muscarininc M 1 receptor agonists as ...